SCHEMBL19902398

SCHEMBL19902398

CCC(=O)c1cn2c(n1)sc1ccccc12

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.45
RET P07949 1/20 0.45
PDGFRB P09619 1/20 0.45
KIT P10721 1/20 0.45
PDGFRA P16234 1/20 0.45
FLT3 P36888 1/20 0.45
CYP2C9 P11712 2/20 0.44
CYP1A2 P05177 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
BRAF P15056 1/20 0.41
RIPK1 Q13546 1/20 0.40
KMT2A Q03164 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454456 0.84 FLT3 (0.47) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL2922603 0.82 GAA (0.53) CYP1A2
SCHEMBL2425146 0.82 CYP2C9 (0.50) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL31290648 0.81 PDGFRA (0.45) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL20518829 0.80 ELANE (0.44) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL20518799 0.80 ALDH1A1 (0.52) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL17452632 0.80 FLT3 (0.47) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL12143505 0.78 CSF1R (0.51) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL20229600 0.78 FLT3 (0.44) CSF1RRETPDGFRBKITPDGFRA
SCHEMBL20518794 0.77 CSF1R (0.45) CSF1RRETPDGFRBKITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed