SCHEMBL19902676

SCHEMBL19902676

CCC(=O)c1cnn2ccc(-c3cnn(C)c3)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 1/20 0.41
BRD4 O60885 1/20 0.41
EPHB3 P54753 1/20 0.41
GSK3B P49841 3/20 0.40
DYRK1A Q13627 3/20 0.40
WNT1 P04628 2/20 0.40
FLT3 P36888 1/20 0.40
NEK2 P51955 1/20 0.40
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
ABL1 P00519 2/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
USP30 Q70CQ3 2/20 0.39
TGFBR1 P36897 2/20 0.39
MARK3 P27448 1/20 0.39
JAK1 P23458 2/20 0.38
JAK3 P52333 2/20 0.38
PRKAB2 O43741 1/20 0.38
CSF1R P07333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454339 0.87 BRD4 (0.53) CREBBPBRD4EPHB3GSK3BDYRK1A
SCHEMBL17438060 0.86 PIM1 (0.47) CREBBPBRD4EPHB3FLT3NEK2
SCHEMBL17452626 0.82 CREBBP (0.43) CREBBPBRD4EPHB3GSK3BDYRK1A
SCHEMBL20229576 0.82 USP30 (0.52) BRD4MKNK1MKNK2USP30MARK3
SCHEMBL25416397 0.74 FLT3 (0.40) DYRK1AFLT3PIM1PIM2MKNK1
SCHEMBL27430475 0.74 PDK2 (0.48) CREBBPBRD4EPHB3ABL1TGFBR1
SCHEMBL3689503 0.74 PIK3CD (0.47) EPHB3
SCHEMBL19997216 0.74 EPHB3 (0.56) EPHB3
SCHEMBL19997277 0.72 ROCK1 (0.50) EPHB3ABL1
SCHEMBL21946562 0.72 FLT3 (0.59) FLT3NEK2ABL1USP30CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed