SCHEMBL19903042

SCHEMBL19903042

COc1cccnc1N1CCN(C(=O)c2cc(C)ccc2-n2nccn2)CCO1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.51
HCRTR2 O43614 18/20 0.47
CYP3A4 P08684 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902988 0.89 HCRTR1 (0.50) HCRTR1HCRTR2CYP3A4
SCHEMBL19903040 0.83 HCRTR1 (0.56) HCRTR1HCRTR2
SCHEMBL19903064 0.82 HCRTR1 (0.52) HCRTR1HCRTR2CYP3A4
SCHEMBL19903009 0.81 HCRTR1 (0.53) HCRTR1HCRTR2
SCHEMBL19903088 0.81 HCRTR2 (0.53) HCRTR1HCRTR2
SCHEMBL19903115 0.81 HCRTR2 (0.64) HCRTR1HCRTR2
SCHEMBL19903005 0.79 HCRTR2 (0.53) HCRTR1HCRTR2CYP3A4
SCHEMBL19903058 0.79 HCRTR2 (0.51) HCRTR1HCRTR2CYP3A4
SCHEMBL19902980 0.79 HCRTR1 (0.49) HCRTR1HCRTR2CYP3A4
SCHEMBL19903099 0.79 HCRTR2 (0.50) HCRTR1HCRTR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3287454-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2020-09-02 EP disclosed
EP-3287454-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2018-02-28 EP disclosed