SCHEMBL19903057

SCHEMBL19903057

Cc1ccccc1-c1cc(Cl)ncc1N(C)C

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 18/20 0.62
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28056546 0.81 GPBAR1 (0.56) GPBAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL12098102 0.78 GPBAR1 (1.00) GPBAR1
SCHEMBL1868987 0.74 CYP1A2 (0.46) GPBAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL1867632 0.74 GPBAR1 (0.69) GPBAR1CYP3A4
SCHEMBL1870080 0.74 GPBAR1 (0.60) GPBAR1CYP3A4
SCHEMBL1876978 0.73 GPBAR1 (0.59) GPBAR1CYP3A4
SCHEMBL12098023 0.73 GPBAR1 (1.00) GPBAR1
SCHEMBL1868986 0.73 GPBAR1 (0.45) GPBAR1CYP1A2CYP3A4CYP2D6
SCHEMBL5555501 0.73 GPBAR1 (0.45) GPBAR1ALDH1A1CYP1A2CYP2C19CYP2C9
SCHEMBL30376925 0.73 GPBAR1 (0.76) GPBAR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3067349-B1 CARBOXYMETHYL PIPERIDINE DERIVATIVE KISSEI PHARMACEUTICAL (JP) 2018-02-28 EP disclosed