SCHEMBL19904657

SCHEMBL19904657

CNC(=O)[C@@H]1CCN(c2ccc3ccccc3c2)C1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 7/20 0.59
PDK2 Q15119 1/20 0.49
ABL1 P00519 1/20 0.46
DPP4 P27487 2/20 0.46
SLC6A9 P48067 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
HTR3A P46098 1/20 0.46
PDE10A Q9Y233 1/20 0.45
MAP4K4 O95819 1/20 0.45
SYK P43405 1/20 0.45
AKR1C3 P42330 2/20 0.43
AKR1C1 Q04828 1/20 0.43
TPSAB1 Q15661 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16695224 0.83 NOTUM (0.69) NOTUMAKR1C3AKR1C1
SCHEMBL16695200 0.83 NOTUM (0.69) NOTUMAKR1C3AKR1C1
SCHEMBL16695072 0.82 DPP4 (0.52) NOTUMPDK2DPP4SLC6A9HTR3A
SCHEMBL29604898 0.82 DPP4 (0.52) NOTUMPDK2DPP4SLC6A9HTR3A
SCHEMBL16695079 0.82 DPP4 (0.52) NOTUMPDK2DPP4SLC6A9HTR3A
SCHEMBL12674885 0.78 NOTUM (0.50) NOTUMPDK2MAP4K4SYK
SCHEMBL19904490 0.78 NOTUM (0.68) NOTUMMAP4K4SYKAKR1C3
SCHEMBL13733384 0.78 NOTUM (0.57) NOTUMPDK2RXFP1MAP4K4SYK
SCHEMBL5799831 0.77 NOTUM (0.55) NOTUMPDK2SLC6A9HTR3AAKR1C3
SCHEMBL12675626 0.77 NOTUM (0.51) NOTUMPDK2ABL1MAP4K4SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed