SCHEMBL19905041

SCHEMBL19905041

CNC(=O)c1ccnc2c(CCNc3cc(-c4ccc(C5(C#N)CC5)cc4)ncn3)cccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 11/20 0.38
CYP3A4 P08684 9/20 0.38
CLK4 Q9HAZ1 9/20 0.38
CYP2C19 P33261 8/20 0.38
ALDH1A1 P00352 8/20 0.38
CYP2D6 P10635 7/20 0.38
USP2 O75604 6/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALOX15 P16050 3/20 0.36
CYP2C9 P11712 2/20 0.36
HSD17B10 Q99714 5/20 0.35
FFAR4 Q5NUL3 1/20 0.34
SCN9A Q15858 2/20 0.34
SLC40A1 Q9NP59 1/20 0.34
LMNA P02545 2/20 0.33
MAPK1 P28482 2/20 0.33
WDR5 P61964 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19355281 0.88 CYP1A2 (0.45) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL19355460 0.86 CYP1A2 (0.44) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL19355476 0.86 FAAH (0.42) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL19355128 0.86 CYP1A2 (0.41) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL17634695 0.85 PRKDC (0.46) SCN9ASLC40A1WDR5PREPFAAH
SCHEMBL19355266 0.84 CYP1A2 (0.43) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL19355473 0.84 CYP1A2 (0.43) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL19355284 0.84 CYP1A2 (0.50) CYP1A2CYP3A4CLK4CYP2C19ALDH1A1
SCHEMBL19355525 0.83 PRKDC (0.39) SCN9ASLC40A1WDR5FAAH
SCHEMBL19355526 0.83 PRKDC (0.39) SCN9ASLC40A1WDR5FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed