SCHEMBL19905084

SCHEMBL19905084

CNC(=O)c1ccnc2c(CCNc3cc(-c4cncc(S(C)(=O)=O)c4)ncn3)cccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 14/20 0.41
CYP3A4 P08684 14/20 0.41
CLK4 Q9HAZ1 11/20 0.41
CYP2C19 P33261 9/20 0.41
CYP2D6 P10635 9/20 0.41
HSD17B10 Q99714 9/20 0.41
ALDH1A1 P00352 7/20 0.41
USP2 O75604 4/20 0.41
ALOX15 P16050 3/20 0.41
SLC40A1 Q9NP59 1/20 0.40
PIK3C3 Q8NEB9 1/20 0.38
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CYP2C9 P11712 2/20 0.36
TSHR P16473 1/20 0.36
KDM4E B2RXH2 2/20 0.35
HPGD P15428 1/20 0.35
NR1H2 P55055 1/20 0.34
MAPK1 P28482 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905163 0.90 SLC40A1 (0.42) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL19355276 0.88 CYP1A2 (0.52) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL20373466 0.87 SLC40A1 (0.39) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL19905409 0.87 CYP1A2 (0.41) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL20373150 0.86 CYP1A2 (0.50) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL19819890 0.86 CYP1A2 (0.45) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL19819893 0.85 CYP1A2 (0.43) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL19355520 0.85 SLC40A1 (0.42) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL17634836 0.84 PRKDC (0.47) CYP1A2CYP3A4CLK4CYP2C19CYP2D6
SCHEMBL19819878 0.84 CYP1A2 (0.40) CYP1A2CYP3A4CLK4CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed