SCHEMBL19905097

SCHEMBL19905097

CNC(=O)c1c(F)cnc2c(C(C)[C@H](C)CNc3cc(-c4cnc(OC)c(OC)c4)ncn3)cccc12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.38
FAAH O00519 5/20 0.38
PIK3CA P42336 8/20 0.36
PIK3CG P48736 7/20 0.36
PIK3CD O00329 2/20 0.36
PIK3CB P42338 1/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2D6 P10635 3/20 0.36
CLK4 Q9HAZ1 3/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GRM7 Q14831 1/20 0.34
USP2 O75604 1/20 0.34
HDAC1 Q13547 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905389 0.94 PRKDC (0.37) PRKDCFAAHPIK3CAPIK3CGPIK3CD
SCHEMBL22838703 0.93 PRKDC (0.37) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL17634849 0.92 PRKDC (0.44) PRKDCFAAHPIK3CAPIK3CGPIK3CD
SCHEMBL19905459 0.92 PRKDC (0.42) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL19905199 0.91 PRKDC (0.38) PRKDCFAAHPIK3CACYP1A2CYP3A4
SCHEMBL19905352 0.89 PRKDC (0.41) PRKDCFAAH
SCHEMBL19905485 0.89 PRKDC (0.42) PRKDCFAAH
SCHEMBL20373310 0.89 PRKDC (0.42) PRKDCFAAH
SCHEMBL19905048 0.88 PRKDC (0.39) PRKDCFAAH
SCHEMBL17634853 0.87 PRKDC (0.42) PRKDCFAAHPIK3CACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed