SCHEMBL19905770

SCHEMBL19905770

Cc1cc2nc(-c3ccnc(-c4cncc(C(=O)O)c4)c3)sc2c(-c2ccc(Cl)cc2)c1C(OC(C)(C)C)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
PSIP1 O75475 1/20 0.34
PSD A5PKW4 1/20 0.32
MAP4K4 O95819 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15341114 1.00 CYP3A4 (0.38) CYP3A4PSIP1PSDMAP4K4
SCHEMBL15340996 0.95 CYP3A4 (0.33) CYP3A4PSDMAP4K4
SCHEMBL15341117 0.94 MAP4K4 (0.37) CYP3A4PSIP1PSDMAP4K4
SCHEMBL15333171 0.91 CYP3A4 (0.37) CYP3A4PSIP1
SCHEMBL15526309 0.91 CYP3A4 (0.37) CYP3A4PSIP1
SCHEMBL20128437 0.89 CYP3A4 (0.39) CYP3A4PSIP1PSD
SCHEMBL15340993 0.89 MAP4K4 (0.37) CYP3A4PSDMAP4K4
SCHEMBL15341098 0.88 CYP3A4 (0.39) CYP3A4PSIP1MAP4K4
SCHEMBL19906063 0.88 CYP3A4 (0.39) CYP3A4PSIP1MAP4K4
SCHEMBL15341121 0.88 PSD (0.40) CYP3A4PSIP1PSDMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed