SCHEMBL19905792

SCHEMBL19905792

Cc1cc2nc(-c3ccnc(-c4ncc5c(n4)c(C)nn5C)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 15/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
PDE5A O76074 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE7A Q13946 1/20 0.32
PDE1C Q14123 1/20 0.32
PDE3A Q14432 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
MAPT P10636 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905921 0.88 KDM4E (0.36) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906076 0.86 KDM4E (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL17530332 0.85
SCHEMBL17530325 0.85
SCHEMBL19906351 0.84 PTGDR2 (0.41) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL15333867 0.83 CYP3A4 (0.38)
SCHEMBL19906023 0.83 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL17547144 0.82 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906178 0.82 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906287 0.82 KDR (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed