SCHEMBL19905935

SCHEMBL19905935

Cc1cc2nc(-c3cnc4c(c3)c(C3=CCN(C)CC3)cn4C)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
WNT1 P04628 2/20 0.33
GSK3B P49841 2/20 0.33
DYRK1A Q13627 2/20 0.33
CLK2 P49760 1/20 0.33
CLK3 P49761 1/20 0.33
KIT P10721 1/20 0.32
HTR1A P08908 1/20 0.32
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CDK4 P11802 1/20 0.31
CCNB1 P14635 1/20 0.31
CCND1 P24385 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
HTR6 P50406 2/20 0.31
EGLN1 Q9GZT9 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20030734 0.93 KDM4E (0.36) KDM4EKMT2AMEN1ALDH1A1WNT1
SCHEMBL19905929 0.90 EIF4EBP1 (0.32) KDM4EKMT2AMEN1ALDH1A1PTGDR2
SCHEMBL15342591 0.84 PSIP1 (0.35)
SCHEMBL22506340 0.84 PSIP1 (0.35)
SCHEMBL19906158 0.84 KDM4E (0.34) KDM4EKMT2AMEN1ALDH1A1PTGDR2
SCHEMBL19905785 0.84 KDM4E (0.38) KDM4EKMT2AMEN1ALDH1A1PTGDR2
SCHEMBL20030685 0.83 KDM4E (0.33) KDM4EKMT2AMEN1ALDH1A1PTGDR2
SCHEMBL31114857 0.83 CNR1 (0.31)
SCHEMBL20101206 0.83 CNR1 (0.31)
SCHEMBL19906364 0.83 KDM4E (0.36) KDM4EKMT2AMEN1ALDH1A1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed