SCHEMBL19905988

SCHEMBL19905988

Cc1cc2nc(-c3cccc(-c4cnc5cnn(C)c5c4)c3)sc2c(-c2ccc(Cl)cc2OC(C)(C)C)c1CC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
MAP4K4 O95819 2/20 0.31
FFAR1 O14842 2/20 0.31
HTT P42858 1/20 0.30
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906320 0.90 KDM4E (0.31) KDM4EPTGDR2MEN1ALDH1A1KMT2A
SCHEMBL19905884 0.88 KDM4E (0.38) KDM4EPTGDR2MEN1ALDH1A1KMT2A
SCHEMBL19906086 0.87 KDM4E (0.39) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19905880 0.86 KDM4E (0.38) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19906060 0.86 KDM4E (0.38) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19906157 0.85 KDM4E (0.38) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19906391 0.83 KDM4E (0.33) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19905850 0.83 KDM4E (0.36) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19906017 0.83 KDM4E (0.32) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1
SCHEMBL19905888 0.83 KDM4E (0.35) KDM4EPTGDR2SMN1; SMN2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed