SCHEMBL19906020

SCHEMBL19906020

Cc1cc2nc(-c3cccc(-c4cnn(CC(C)C)c4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
S1PR1 P21453 1/20 0.36
LIPC P11150 1/20 0.36
PTGDR2 Q9Y5Y4 4/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PFKFB3 Q16875 1/20 0.35
NAMPT P43490 1/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
SOS1 Q07889 1/20 0.33
JAK2 O60674 1/20 0.33
KLKB1 P03952 1/20 0.33
PDK2 Q15119 1/20 0.33
PDE5A O76074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905831 0.90 PIK3CD (0.42) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9
SCHEMBL19905796 0.89 KDM4E (0.39) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9
SCHEMBL19905882 0.88 KDM4E (0.41) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9
SCHEMBL19906018 0.88 KDM4E (0.35) KDM4ES1PR1LIPCPTGDR2ALDH1A1
SCHEMBL17547146 0.85 KDM4E (0.39) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9
SCHEMBL15341113 0.84 CYP3A4 (0.37) S1PR1LIPC
SCHEMBL17547045 0.83 KDM4E (0.37) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9
SCHEMBL15341043 0.82 LIPC (0.36) S1PR1LIPCPFKFB3NAMPTPRMT5
SCHEMBL19906088 0.81 KDM4E (0.42) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9
SCHEMBL19905803 0.81 KDM4E (0.39) KDM4EPTGDR2ALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed