SCHEMBL19906047

SCHEMBL19906047

Cc1cc2nc(-c3ccnc(-c4ccc5ccn(C)c(=O)c5c4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.35
PTGDR2 Q9Y5Y4 7/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
AKR1B1 P15121 3/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
MCHR1 Q99705 1/20 0.32
CASP3 P42574 1/20 0.31
SENP8 Q96LD8 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
BRD4 O60885 1/20 0.30
KDM5A P29375 1/20 0.30
KDM4C Q9H3R0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906103 0.92 MCHR1 (0.33) KDM4EROCK2ROCK1MCHR1CASP3
SCHEMBL19906102 0.89 KDM4E (0.32) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905816 0.87 KDM4E (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906265 0.86 KDM4E (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905985 0.85 KDM4E (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906277 0.85 PTGDR2 (0.37) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905917 0.84 PTGDR2 (0.38) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906076 0.84 KDM4E (0.37) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905872 0.84 PTGDR2 (0.37) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL17547144 0.84 PTGDR2 (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed