SCHEMBL19906103

SCHEMBL19906103

CCc1c(C)cc2nc(-c3ccnc(-c4ccc5ccn(C)c(=O)c5c4)c3)sc2c1-c1ccc(Cl)cc1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.33
SREBF2 Q12772 1/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.32
BRD4 O60885 1/20 0.32
CASP3 P42574 1/20 0.30
SENP8 Q96LD8 1/20 0.30
SENP7 Q9BQF6 1/20 0.30
SENP6 Q9GZR1 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906047 0.92 KDM4E (0.35) MCHR1KDM4EBRD4CASP3SENP8
SCHEMBL19906102 0.81 KDM4E (0.32) KDM4ELMNA
SCHEMBL15342248 0.81
SCHEMBL15342668 0.81 CYP3A4 (0.35)
SCHEMBL19906065 0.79 SREBF2 (0.35) SREBF2KDM4ELMNAMAPTATM
SCHEMBL19905816 0.78 KDM4E (0.35) MCHR1KDM4EIDH1
SCHEMBL19906265 0.77 KDM4E (0.35) SREBF2KDM4ECASP3SENP8SENP7
SCHEMBL19905985 0.77 KDM4E (0.35) MCHR1KDM4EMAPTIDH1
SCHEMBL19906277 0.76 PTGDR2 (0.37) KDM4ENPC1RAB9A
SCHEMBL19906076 0.75 KDM4E (0.37) MCHR1KDM4ELMNAMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed