SCHEMBL19906310

SCHEMBL19906310

Cc1cc2nc(-c3cncc(-c4ccc5c(c4)ncn5C)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
PTGDR2 Q9Y5Y4 7/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GFER P55789 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
WNT1 P04628 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
MCHR1 Q99705 1/20 0.32
MCL1 Q07820 1/20 0.31
PDE5A O76074 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906198 0.93 NPC1 (0.40) NPC1RAB9ASMN1; SMN2TP53PTGDR2
SCHEMBL19905758 0.86 PTGDR2 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL15341123 0.81 CYP3A4 (0.39) NPC1RAB9ASMN1; SMN2TP53
SCHEMBL19906197 0.81 PTGDR2 (0.36) NPC1RAB9ASMN1; SMN2TP53PTGDR2
SCHEMBL19906233 0.81 PTGDR2 (0.34) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905939 0.80 PTGDR2 (0.35) NPC1RAB9ASMN1; SMN2PTGDR2KDM4E
SCHEMBL19906327 0.80 PTGDR2 (0.38) NPC1RAB9ASMN1; SMN2PTGDR2KDM4E
SCHEMBL19906180 0.80 PTGDR2 (0.41) NPC1RAB9ASMN1; SMN2PTGDR2KDM4E
SCHEMBL15340998 0.80 NPC1 (0.33) NPC1RAB9ASMN1; SMN2TP53GFER
SCHEMBL19905876 0.80 PTGDR2 (0.42) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed