SCHEMBL19908368

SCHEMBL19908368

CC1(C)CCc2cccnc2CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.40
GRIN2B Q13224 4/20 0.40
DRD2 P14416 2/20 0.39
DRD3 P35462 1/20 0.39
IDH1 O75874 3/20 0.32
SIGMAR1 Q99720 2/20 0.31
CYP2D6 P10635 2/20 0.31
CNR2 P34972 1/20 0.31
NAMPT P43490 1/20 0.30
AKR1C3 P42330 1/20 0.30
CHRM2 P08172 1/20 0.30
HTR1A P08908 1/20 0.30
CHRM1 P11229 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
ADRA1A P35348 1/20 0.30
HRH1 P35367 1/20 0.30
OPRK1 P41145 1/20 0.30
HTR2B P41595 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708059 0.87 CNR2 (0.38) GRIN1GRIN2BDRD2DRD3IDH1
SCHEMBL30667082 0.87 DRD2 (0.38) GRIN1GRIN2BDRD2DRD3IDH1
SCHEMBL11418045 0.87 DRD2 (0.38) GRIN1GRIN2BDRD2DRD3IDH1
SCHEMBL17413659 0.77 DRD2 (0.42) GRIN1GRIN2BDRD2DRD3IDH1
SCHEMBL8348677 0.77
Hydrochloric Acid SCHEMBL8777224 0.74 DRD2 (0.41) GRIN1GRIN2BDRD2DRD3IDH1
Bromide SCHEMBL8777272 0.74 DRD2 (0.41) GRIN1GRIN2BDRD2DRD3IDH1
SCHEMBL9418958 0.74 TSHR (0.48) DRD2DRD3SIGMAR1HTR2AHTR2C
Trifluoromethanesulfonic Acid SCHEMBL28119326 0.73 CNR2 (0.38) IDH1CNR2NAMPT
SCHEMBL20840517 0.73 DRD2 (0.36) GRIN1GRIN2BDRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191483-B1 COMPOUNDS AS CRTH2 ANTAGONIST AND USES THEREOF NORTH & SOUTH BROTHER PHARMACY INVESTMENT CO LTD (CN) 2020-06-10 EP disclosed
EP-3287461-A1 IMIDAZO ISOINDOLE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Jiangsu Hengrui Medicine Co., Ltd. (CN) 2018-02-28 EP disclosed