SCHEMBL19908474

SCHEMBL19908474

CC1(C)Nc2ncc(-c3ccc(C(=O)N4CCCC4)cc3)cc2N(Cc2cc(F)ccc2F)C1=O

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 7/20 0.54
RIPK1 Q13546 3/20 0.43
NTRK1 P04629 5/20 0.42
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
MAPT P10636 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
ROCK2 O75116 1/20 0.37
GRIN2B Q13224 1/20 0.36
ENPP2 Q13822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1600425 0.94 NTRK1 (0.49) ALKRIPK1NTRK1ALDH1A1HTT
SCHEMBL14387471 0.87 ALK (0.59) ALKNTRK1HPGD
SCHEMBL1601019 0.86 ALK (0.76) ALK
SCHEMBL1601018 0.86 ALK (0.76) ALK
SCHEMBL19908262 0.84 ALK (0.54) ALKRIPK1NTRK1ALDH1A1HTT
SCHEMBL1602277 0.78 ALK (0.66) ALKNTRK1
SCHEMBL19908264 0.78 AR (0.38) ALKNTRK1ALDH1A1ROCK2
SCHEMBL1601642 0.78 ALK (0.51) ALKRIPK1NTRK1
SCHEMBL1602786 0.77 AR (0.37) ALKNTRK1ROCK2
SCHEMBL1600401 0.77 ALK (0.70) ALKNTRK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091951-B1 PYRIDO[2,3-B]PYRAZINE AND [1,8]-NAPHTHYRIDINE DERIVATIVES AS ALK AND C-MET INHIBITORS CEPHALON INC (US) 2018-02-28 EP disclosed