SCHEMBL19909277

SCHEMBL19909277

CC1=C(c2cnc(Nc3cccc(N4CCOCC4)c3)nc2)NC1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
CCNT1 O60563 5/20 0.51
CDK2 P24941 5/20 0.51
CDK9 P50750 5/20 0.51
CCNE1 P24864 1/20 0.51
CCNA2 P20248 4/20 0.49
CDK1 P06493 1/20 0.48
CCNB1 P14635 1/20 0.48
CDK7 P50613 1/20 0.48
CCNH P51946 1/20 0.48
CCNA1 P78396 1/20 0.48
RIPK2 O43353 2/20 0.47
JAK2 O60674 2/20 0.47
NTRK1 P04629 1/20 0.47
JAK1 P23458 1/20 0.46
JAK3 P52333 1/20 0.46
TTBK1 Q5TCY1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22990854 0.75 CDK2 (0.51) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL5502283 0.74 HDAC3 (0.58) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL519704 0.72 HDAC3 (0.58) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL29371274 0.71 CDK2 (0.62) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL12614697 0.71 HDAC3 (0.64) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL4730099 0.70 HDAC6 (1.00) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL20516550 0.69 RIPK2 (0.71) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL18376719 0.69 MAP4K1 (0.62) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL15824558 0.69 HDAC3 (0.59) HDAC3HDAC1HDAC2HDAC6CCNT1
SCHEMBL17465885 0.68 DCLK1 (0.72) RIPK2PLK4BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935248-B1 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC (US) 2018-02-28 EP disclosed