SCHEMBL19909663

SCHEMBL19909663

CC#CC(=O)N1CC2(CNC2)C1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPX4 P36969 1/20 0.33
BTK Q06187 8/20 0.32
NAMPT P43490 1/20 0.31
NSD2 O96028 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19909717 0.77 GPX4 (0.33) GPX4BTKNSD2
SCHEMBL16122876 0.76 BTK (0.38) BTK
SCHEMBL16078763 0.74 GPX4 (0.37) GPX4BTK
SCHEMBL16075248 0.74 BTK (0.33) GPX4BTK
SCHEMBL2593681 0.73 SMN1; SMN2 (0.45) NAMPT
SCHEMBL30059414 0.72 NAMPT (0.36) NAMPT
SCHEMBL16075032 0.72 BTK (0.42) GPX4BTK
SCHEMBL15472834 0.72 BTK (0.39) BTK
Hydrochloric Acid SCHEMBL16454452 0.71 SMN1; SMN2 (0.43) NAMPT
SCHEMBL2239249 0.70 NAMPT (0.36) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970163-B1 5-THIAZOLECARBOXAMIDE DERVATIVES AND THEIR USE AS BTK INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-02-28 EP disclosed