SCHEMBL19909694

SCHEMBL19909694

CC/C=C(/C(N)=O)C(F)(F)F

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FAAH O00519 8/20 0.31
GRIK1 P39086 1/20 0.31
GRIK2 Q13002 1/20 0.31
CES1 P23141 5/20 0.30
CES2 O00748 2/20 0.30
MEN1 O00255 1/20 0.30
CYP1A2 P05177 1/20 0.30
KMT2A Q03164 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852706 0.79 GRIK1 (0.35) FAAHGRIK1GRIK2CES1CES2
SCHEMBL2852703 0.79 GRIK1 (0.35) FAAHGRIK1GRIK2CES1CES2
SCHEMBL13560398 0.75 TDP1 (0.30)
SCHEMBL13560395 0.75 TDP1 (0.30)
SCHEMBL27757791 0.74 MAPT (0.41) MEN1KMT2A
SCHEMBL27576280 0.72 NPSR1 (0.39) CES1CES2MEN1CYP1A2KMT2A
SCHEMBL28251374 0.71
SCHEMBL11110589 0.70
SCHEMBL25078268 0.70
SCHEMBL8661877 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970163-B1 5-THIAZOLECARBOXAMIDE DERVATIVES AND THEIR USE AS BTK INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-02-28 EP disclosed