SCHEMBL19915938

SCHEMBL19915938

Bc1ccc2cncn2c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 15/20 0.39
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
PTGIS Q16647 1/20 0.38
IDO1 P14902 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19915935 0.81 IDO1 (0.39) TBXAS1IDO1
SCHEMBL21060548 0.79 TBXAS1 (0.39) TBXAS1PTGS1PTGS2PTGISIDO1
SCHEMBL19915855 0.76 IDO1 (0.55) TBXAS1PTGS1PTGS2PTGISIDO1
SCHEMBL21060532 0.72 IDO1 (0.50) TBXAS1PTGS1PTGS2PTGISIDO1
SCHEMBL21816313 0.69 TBXAS1 (0.39) TBXAS1PTGS1PTGS2PTGISIDO1
SCHEMBL5792448 0.68 TBXAS1 (0.51) TBXAS1PTGS1PTGS2PTGISIDO1
SCHEMBL19915857 0.65 IDO1 (0.39) TBXAS1IDO1
SCHEMBL19915741 0.62 IDO1 (0.48) TBXAS1PTGS1PTGS2PTGISIDO1
SCHEMBL18137410 0.62 TBXAS1 (0.44) TBXAS1
SCHEMBL11041767 0.61 TBXAS1 (0.67) TBXAS1PTGS1PTGS2PTGIS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018036414-A1 FUSED HETEROCYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 北京诺诚健华医药科技有限公司 2018-03-01 WO disclosed