SCHEMBL19916769

SCHEMBL19916769

CC(C)(COc1cccc(C(=O)Nc2ccc(Cl)c(-c3ccccn3)c2)c1)C(C)(C)C(=O)NO

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.47
HTR1A P08908 1/20 0.47
SLC6A2 P23975 1/20 0.47
PDE4A P27815 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
HTR2B P41595 1/20 0.47
SLC6A3 Q01959 1/20 0.47
PDE4D Q08499 1/20 0.47
SHH Q15465 1/20 0.47
USP28 Q96RU2 1/20 0.47
SLC29A1 Q99808 1/20 0.47
SMO Q99835 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
MAPT P10636 3/20 0.45
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19916728 0.92 ALB (0.48) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL19916704 0.83 MAPT (0.70) MAPTLMNAGAAHTT
SCHEMBL15424158 0.81 MAPT (0.49) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL19685469 0.81 ALB (0.48) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL19132578 0.81 NR1H4 (0.60) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL15424150 0.79 ALB (0.58) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL2619398 0.76 ALB (0.58) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL15424139 0.76 ALB (0.59) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL28386672 0.76 ALB (0.64) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL19132583 0.75 USP28 (0.59) ALBHTR1ASLC6A2PDE4AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2661425-B1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES CURIS INC (US) 2018-02-28 EP disclosed