SCHEMBL19917243

SCHEMBL19917243

CC(=O)CNC(=O)c1ncc2nc(-c3ccc4ccccc4c3)ccc2c1O

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 11/20 0.52
FTO Q9C0B1 2/20 0.50
EGLN3 Q9H6Z9 1/20 0.50
EGLN2 Q96KS0 10/20 0.46
THRA P10827 2/20 0.40
THRB P10828 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19895134 0.91 EGLN1 (0.63) EGLN1FTOEGLN3EGLN2THRA
SCHEMBL22369548 0.90 EGLN1 (0.47) EGLN1FTOEGLN3EGLN2
SCHEMBL22369546 0.86 EGLN1 (0.45) EGLN1FTOEGLN3EGLN2
SCHEMBL19895129 0.82 ALPL (0.48) EGLN1FTOEGLN3
SCHEMBL22369556 0.80 EGLN1 (0.47) EGLN1FTOEGLN3
SCHEMBL20109765 0.79 EGLN1 (0.67) EGLN1FTOEGLN3EGLN2THRA
SCHEMBL19917277 0.78 EGLN1 (0.61) EGLN1FTOEGLN3THRATHRB
SCHEMBL20109775 0.77 EGLN1 (0.62) EGLN1FTOTHRATHRB
SCHEMBL20109769 0.76 EGLN1 (0.60) EGLN1FTOEGLN2THRATHRB
SCHEMBL25934727 0.76 EGLN1 (0.54) EGLN1FTOEGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3287456-A1 COMPOUND OF 5-HYDROXYL-1,7-NAPHTHYRIDINE SUBSTITUTED BY ARYL OR HETEROARYL, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE THEREOF Shenyang Sunshine Pharmaceutical Co., Ltd. (CN) 2018-02-28 EP disclosed