SCHEMBL19928546

SCHEMBL19928546

CC(CCCN1CCC2(CC1)COC2)N1CCC2(CC1)CNC2

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19928539 0.87 MEN1 (0.31)
SCHEMBL24688458 0.76 OPRM1 (0.32)
SCHEMBL20153166 0.76 TSHR (0.33) TSHR
SCHEMBL21153226 0.74 TOP2A (0.39)
SCHEMBL21160556 0.73 MEN1 (0.33)
SCHEMBL18842878 0.73 TSHR (0.35) TSHR
SCHEMBL22414444 0.71 USP2 (0.31) CYP2D6TSHR
SCHEMBL13766677 0.71 TSHR (0.40) CYP2D6TSHR
SCHEMBL29325143 0.71 CYP2D6 (0.36) CYP1A2CYP2D6
SCHEMBL20921362 0.69 S1PR1 (0.44) CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9908886-B2 Bicyclic heterocyclic derivatives as MNK1 and MNK2 modulators and uses thereof AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-03-06 US disclosed