SCHEMBL19940290

SCHEMBL19940290

COC(=O)c1ccc(C2=CCN(C(=O)OC(C)(C)C)CC2)cc1N

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.53
PDK4 Q16654 1/20 0.47
CDK7 P50613 1/20 0.46
CDK13 Q14004 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
GRM1 Q13255 8/20 0.46
GRM5 P41594 7/20 0.46
LIPC P11150 1/20 0.45
LIPG Q9Y5X9 1/20 0.45
CYP11B2 P19099 1/20 0.44
TNK2 Q07912 1/20 0.43
QDPR P09417 2/20 0.43
SOS1 Q07889 1/20 0.43
JAK1 P23458 1/20 0.43
BTK Q06187 1/20 0.43
NR1H2 P55055 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24718282 0.90 NAMPT (0.56) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL30798377 0.90 NAMPT (0.56) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL3033965 0.88 NAMPT (0.54) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL30736648 0.88 NAMPT (0.54) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL15380388 0.87 NAMPT (0.53) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL30798334 0.87 NAMPT (0.53) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL29152538 0.87 NAMPT (0.53) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL31612866 0.87 NAMPT (0.53) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL16992228 0.87 QDPR (0.54) NAMPTPDK4CDK7CDK13CDK12
SCHEMBL15157008 0.87 NAMPT (0.56) NAMPTPDK4CDK7CDK13CDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018041248-A1 BCL-2 SELECTIVE INHIBITOR AND PREPARATION AND USE THEREOF 北京赛林泰医药技术有限公司 2018-03-08 WO disclosed