SCHEMBL19940563

SCHEMBL19940563

O=C(C(=O)N1CCC[C@H](c2cccc(-c3nc(-n4ccnn4)c4[nH]cc(C(=O)C(=O)N5CCCC(c6ccc(Cl)cc6)C5)c4c3F)c2)C1)c1c[nH]c2c(-n3ccnn3)ncc(F)c12

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 14/20 0.35
BTK Q06187 4/20 0.33
MAPK1 P28482 1/20 0.32
AOC3 Q16853 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16135269 0.89 PROKR1 (0.41) PROKR1
SCHEMBL16135262 0.85 BTK (0.39) BTK
SCHEMBL16135264 0.85 CYP3A4 (0.39) PROKR1
SCHEMBL16135261 0.82 CYP3A4 (0.40)
SCHEMBL16135243 0.80 CYP3A4 (0.40)
SCHEMBL13116885 0.77 MAPT (0.38) BTK
SCHEMBL16135265 0.74 GABRA1 (0.41)
SCHEMBL13116854 0.72 CYP3A4 (0.40)
SCHEMBL13117259 0.72 CYP3A4 (0.39)
SCHEMBL15273565 0.72 CYP3A4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2978763-B1 2-KETO AMIDE DERIVATIVES AS HIV ATTACHMENT INHIBITORS VIIV HEALTHCARE UK (NO 5) LTD (GB) 2018-03-07 EP disclosed