SCHEMBL19946124

SCHEMBL19946124

Cc1nccc2c3ccc(OC[C@@H](C)CC(C)(C)NC(=O)O)cc3c(=O)n(C)c12

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 15/20 0.65
DYRK1A Q13627 4/20 0.42
MAOA P21397 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19946123 0.85 AAK1 (0.84) AAK1DYRK1A
SCHEMBL19946141 0.85 AAK1 (0.61) AAK1
SCHEMBL16972637 0.84 AAK1 (0.47) AAK1DYRK1AMAOA
SCHEMBL21018876 0.83 AAK1 (0.66) AAK1DYRK1AMAOABCHEACHE
SCHEMBL19946030 0.82 AAK1 (0.62) AAK1
SCHEMBL15562280 0.82 AAK1 (0.49) AAK1DYRK1A
SCHEMBL15562155 0.81 AAK1 (0.52) AAK1DYRK1A
SCHEMBL21019088 0.81 AAK1 (0.63) AAK1DYRK1AMAOABCHEACHE
SCHEMBL19946110 0.81 AAK1 (0.62) AAK1DYRK1AMAOA
SCHEMBL21018881 0.79 AAK1 (0.69) AAK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3292124-A2 FUSED PYRIDINES AS ADAPTOR ASSOCIATED KINASE 1 (AAK1) INHIBITORS Bristol-Myers Squibb Company (US) 2018-03-14 EP disclosed