SCHEMBL19946141

SCHEMBL19946141

C[C@H](COc1ccc2c(c1)c(=O)n(C)c1cnccc21)CC(C)(C)NC(=O)O

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 13/20 0.61
ROCK2 O75116 7/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15562155 0.93 AAK1 (0.52) AAK1ROCK2
SCHEMBL19946030 0.88 AAK1 (0.62) AAK1ROCK2
SCHEMBL19946124 0.85 AAK1 (0.65) AAK1
SCHEMBL19946177 0.85 AAK1 (0.71) AAK1ROCK2
SCHEMBL16972637 0.83 AAK1 (0.47) AAK1
SCHEMBL15562077 0.79 AAK1 (0.51) AAK1ROCK2
SCHEMBL15455689 0.78 AAK1 (0.61) AAK1ROCK2
SCHEMBL20176303 0.77 AAK1 (0.75) AAK1
SCHEMBL15562104 0.77 AAK1 (0.55) AAK1ROCK2
SCHEMBL15562193 0.77 AAK1 (0.50) AAK1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3292124-A2 FUSED PYRIDINES AS ADAPTOR ASSOCIATED KINASE 1 (AAK1) INHIBITORS Bristol-Myers Squibb Company (US) 2018-03-14 EP disclosed