SCHEMBL19946331

SCHEMBL19946331

CC(C)(C)OC(=O)NOC(=O)Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.48
PPARA Q07869 1/20 0.48
MAPK8 P45983 2/20 0.45
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
MAPK10 P53779 1/20 0.40
PIK3CA P42336 1/20 0.40
RXRA P19793 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NLRP3 Q96P20 1/20 0.39
CNR2 P34972 1/20 0.39
LTA4H P09960 1/20 0.38
EPHX2 P34913 1/20 0.38
IDO1 P14902 2/20 0.38
MAOB P27338 2/20 0.38
CYP17A1 P05093 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19946326 0.84 MAPK8 (0.49) PPARGPPARAMAPK8SMN1; SMN2NLRP3
SCHEMBL1948655 0.82 CA12 (0.50) PPARGPPARASMN1; SMN2IDO1
SCHEMBL1948560 0.81 HDAC1 (0.41) PPARGPPARAHDAC1MAPTSMN1; SMN2
SCHEMBL27739636 0.79 PPARG (0.46) PPARGPPARAMAPK8HDAC1HDAC8
SCHEMBL30678949 0.78 HDAC1 (0.41) PPARGPPARAMAPK8HDAC1HDAC8
SCHEMBL13595526 0.78 PPARG (0.48) PPARGPPARALMNAMAPT
SCHEMBL841124 0.77 CYP4F2 (0.58) MAPK8HDAC1HDAC8MAPK10PIK3CA
SCHEMBL4574985 0.77 LSS (0.52) PPARGPPARAHDAC1HDAC8EPHX2
SCHEMBL4655026 0.76 CA12 (0.44) PPARGPPARAMAPTSMN1; SMN2
SCHEMBL7739224 0.76 NR1H2 (0.40) PPARGPPARANR1H2NR1H3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2848618-B1 NITROGENATED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2018-03-14 EP disclosed