SCHEMBL19953049

SCHEMBL19953049

Clc1ccc(-n2cncc2-c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.58
CYP11B2 P19099 4/20 0.58
CRBN Q96SW2 1/20 0.48
HSP90AA1 P07900 2/20 0.48
HSP90AB1 P08238 2/20 0.48
IDO1 P14902 2/20 0.47
CYP1A2 P05177 1/20 0.42
LDLR P01130 1/20 0.42
PCSK9 Q8NBP7 1/20 0.42
FGFR1 P11362 1/20 0.41
LMNA P02545 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GRM1 Q13255 1/20 0.41
FLT3 P36888 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12676747 0.87 CYP11B1 (0.50) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1
SCHEMBL19953122 0.83 HSP90AA1 (0.46) CYP11B1CYP11B2HSP90AA1HSP90AB1LMNA
SCHEMBL11394015 0.83 CRBN (0.48) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1
SCHEMBL12685600 0.82 IDO1 (0.49) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1
SCHEMBL27989267 0.80 CYP11B1 (0.48) CYP11B1CYP11B2HSP90AA1HSP90AB1IDO1
SCHEMBL19953112 0.80 CRBN (0.53) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1
SCHEMBL27836638 0.79 CRBN (0.45) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1
SCHEMBL11384012 0.79 CYP11B1 (0.59) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1
SCHEMBL6291198 0.77 PTGS2 (0.60) IDO1
SCHEMBL27989478 0.77 CYP11B1 (0.49) CYP11B1CYP11B2CRBNHSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed
CN-1178938-C 1,2-annelated quinoline derivatives ղɭҩҵ���޹�˾ 2004-12-08 CN disclosed
CN-1331693-A 1,2-annelated quinoline derivatives JANSSEN PHARMACEUTICA NV (BE) 2002-01-16 CN disclosed