SCHEMBL19953203

SCHEMBL19953203

Cc1cc(F)c(-c2cnc(Cl)n2-c2ccc(Cl)cc2)c(F)c1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.43
PTGS1 P23219 2/20 0.42
POLB P06746 1/20 0.41
AOC3 Q16853 3/20 0.40
KCNH2 Q12809 3/20 0.40
PIK3CA P42336 1/20 0.36
NOTUM Q6P988 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110782 0.80 PTGS2 (0.44) PTGS2POLBAOC3KCNH2PIK3CA
SCHEMBL19953110 0.77 PTGS2 (0.40) PTGS2PTGS1AOC3KCNH2
SCHEMBL1110963 0.75 PTGS2 (0.44) PTGS2AOC3KCNH2PIK3CA
SCHEMBL1074708 0.75 PTGS2 (0.42) PTGS2AOC3KCNH2PIK3CAKDM4E
SCHEMBL19953171 0.74 POLB (0.41) POLBAOC3KCNH2NOTUMKDM4E
SCHEMBL19953079 0.74 HSP90AA1 (0.48) POLBAOC3KCNH2
SCHEMBL19953198 0.73 PTGS2 (0.68) PTGS2PTGS1AOC3KCNH2PIK3CA
SCHEMBL19953204 0.69 PTGS2 (0.49) PTGS2AOC3KCNH2ALDH1A1
SCHEMBL1075327 0.68 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL2450998 0.67 PTGS2 (0.40) PTGS2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed