SCHEMBL19953631

SCHEMBL19953631

COC(=O)C1C(=O)N(C)Cc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
TSHR P16473 1/20 0.40
XIAP P98170 1/20 0.40
BRD4 O60885 2/20 0.38
CREBBP Q92793 1/20 0.38
MMP2 P08253 1/20 0.37
ANPEP P15144 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
POLB P06746 1/20 0.36
PARP1 P09874 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953500 0.79 FABP5 (0.44) HDAC4HDAC7HDAC5TSHRXIAP
SCHEMBL1207850 0.76 HDAC4 (0.51) HDAC4HDAC7HDAC5TSHRANPEP
SCHEMBL5400138 0.76 CHRM2 (0.45) HDAC4HDAC7HDAC5TSHRXIAP
SCHEMBL26730530 0.75 PDE4A (0.41) TSHRXIAP
SCHEMBL22861976 0.74 BRD4 (0.45) TSHRBRD4CREBBPCHRM2CHRM1
SCHEMBL4989954 0.72 ANPEP (0.50) TSHRXIAPBRD4CREBBPANPEP
Hydrochloric Acid SCHEMBL22612124 0.71 ANPEP (0.51) XIAPBRD4CREBBPANPEPPARP1
Hydrochloric Acid SCHEMBL30630763 0.71 ANPEP (0.51) XIAPBRD4CREBBPANPEPPARP1
SCHEMBL20777955 0.71 HDAC4 (0.36) HDAC4HDAC7HDAC5TSHRPOLB
SCHEMBL8804810 0.71 HSD17B10 (0.41) HDAC4HDAC7HDAC5TSHRSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed