SCHEMBL19954200

SCHEMBL19954200

CCC(C)(CC)NCC(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.51
MAPK1 P28482 1/20 0.47
ALDH1A1 P00352 2/20 0.47
POLB P06746 1/20 0.47
ADRB2 P07550 1/20 0.46
ADRB1 P08588 1/20 0.46
ADRB3 P13945 1/20 0.46
CES1 P23141 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
MMP8 P22894 1/20 0.45
PKM P14618 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2294639 0.86 ADRB2 (0.56) GSK3BMAPK1ALDH1A1ADRB2ADRB1
SCHEMBL2293183 0.78 GSK3B (0.57) GSK3BMAPK1ALDH1A1POLBCES1
SCHEMBL255269 0.78 GSK3B (0.61) GSK3BMAPK1ALDH1A1CES1NPC1
SCHEMBL671514 0.76 GSK3B (0.67) GSK3BMAPK1ALDH1A1CES1CA1
SCHEMBL4472065 0.75 SMN1; SMN2 (0.58) GSK3BMAPK1ALDH1A1CES1NPC1
SCHEMBL1699076 0.75 GSK3B (0.57) GSK3BMAPK1ALDH1A1ADRB2ADRB1
SCHEMBL11510574 0.75 GSK3B (0.71) GSK3BMAPK1ALDH1A1POLBCES1
SCHEMBL255479 0.74 GSK3B (0.61) GSK3BMAPK1ALDH1A1POLBCES1
SCHEMBL14041426 0.74 GSK3B (0.61) GSK3BMAPK1ALDH1A1CES1CA1
SCHEMBL23728041 0.74 PPARG (0.49) GSK3BMAPK1ALDH1A1ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9914740-B2 Tricyclic pyrido-carboxamide derivatives as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2018-03-13 US disclosed