SCHEMBL19954223

SCHEMBL19954223

Cc1cc(CNN(C)C)no1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.42
PDE10A Q9Y233 1/20 0.40
MAPT P10636 3/20 0.38
RECQL P46063 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
ALDH1A1 P00352 1/20 0.35
EGFR P00533 1/20 0.35
GAA P10253 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTR2A P28223 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4156491 0.78
SCHEMBL22593293 0.78
SCHEMBL18868074 0.76
SCHEMBL2259618 0.74 EPHX2 (0.43) EPHX2PDE10AMAPTRECQLTRPM8
SCHEMBL18270145 0.74 MAPT (0.41) EPHX2PDE10AMAPTRECQLTRPM8
SCHEMBL12062404 0.73 EPHX2 (0.42) EPHX2PDE10AMAPTRECQLTRPM8
SCHEMBL104242 0.73 TRPM8 (0.50) EPHX2PDE10AMAPTRECQLTRPM8
SCHEMBL3750450 0.72 EPHX2 (0.44) EPHX2PDE10AMAPTRECQLTRPM8
SCHEMBL2755867 0.72 EPHX2 (0.58) EPHX2PDE10AMAPTNPC1RAB9A
SCHEMBL14724572 0.72 EPHX2 (0.41) EPHX2PDE10AMAPTRECQLTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9914740-B2 Tricyclic pyrido-carboxamide derivatives as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2018-03-13 US disclosed