SCHEMBL19956734

SCHEMBL19956734

c1ncc2ncn(-c3ccc(C4CCCCC4)cc3)c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 1/20 0.46
DGAT1 O75907 2/20 0.40
CYP11B2 P19099 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ATM Q13315 1/20 0.37
ALDH1A1 P00352 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
PI4KA P42356 2/20 0.34
PI4K2B Q8TCG2 2/20 0.34
PI4K2A Q9BTU6 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13190252 0.79 DGAT1 (0.68) MKNK2DGAT1ALDH1A1CYP1A2CYP2C19
SCHEMBL19956781 0.79 DGAT1 (0.68) MKNK2DGAT1ALDH1A1CYP1A2CYP2C19
SCHEMBL13190441 0.76 DGAT1 (0.65) DGAT1PI4KAPI4K2BPI4K2API4KB
SCHEMBL13190315 0.76 PI4KA (0.62) DGAT1KMT2ASMN1; SMN2TDP1ALDH1A1
SCHEMBL3697841 0.76 MKNK2 (0.49) MKNK2KMT2ASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL680855 0.75 FGFR1 (0.56) MKNK2HTTKMT2AALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL4456679 0.73 FGFR1 (0.54) MKNK2HTTKMT2AALDH1A1CYP1A2
SCHEMBL467133 0.72 MKNK2 (0.47) MKNK2HTTKMT2AALDH1A1CYP1A2
SCHEMBL28839763 0.71 MKNK2 (0.43) MKNK2KMT2AALDH1A1CYP1A2CYP2C19
SCHEMBL28317574 0.70 MKNK2 (0.55) MKNK2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805951-B1 Inhibitors of diacylglycerol o-acyltransferase 1 (DGAT-1) and uses thereof METABASIS THERAPEUTICS INC (US) 2018-03-14 EP disclosed