SCHEMBL19964465

SCHEMBL19964465

NCc1cc2occc2s1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.47
ASIC3 Q9UHC3 1/20 0.47
LOXL2 Q9Y4K0 1/20 0.47
HTR1B P28222 2/20 0.31
CYP2E1 P05181 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2B6 P20813 1/20 0.31
CYP2C19 P33261 1/20 0.31
LOX P28300 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5039451 0.79 CYP2A6 (0.47) CYP2A6HTR1B
SCHEMBL5036056 0.78
SCHEMBL5039863 0.76 CYP2A6 (0.32) CYP2A6
SCHEMBL5039591 0.74
SCHEMBL5036768 0.69 KMT2A (0.34) CYP3A4
SCHEMBL5035904 0.69 KDM4E (0.36) CYP2A6CYP3A4CYP2C9CYP2C19
SCHEMBL17104854 0.69 ALDH1A1 (0.30)
SCHEMBL13032428 0.65 CYP2A6 (0.45) CYP2A6ASIC3LOXL2CA2
SCHEMBL1253252 0.64 CYP2A6 (0.47) CYP2A6ASIC3LOXL2CYP2E1CYP3A4
SCHEMBL17080670 0.64 CYP2A6 (0.58) CYP2A6ASIC3LOXL2CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048930-A1 LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA, INC. (US) 2018-03-15 WO disclosed