SCHEMBL19965760

SCHEMBL19965760

CCc1nc2c(s1)N(C1COC1)CC2

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.31
RECQL P46063 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14930326 0.80 PDE10A (0.30)
SCHEMBL21769131 0.79
SCHEMBL14925538 0.77
SCHEMBL23109923 0.74 RAD52 (0.40) RAD52RECQLGRM5
SCHEMBL12344027 0.74 GRM5 (0.37) RAD52RECQLGRM5
SCHEMBL19965759 0.71 GRM5 (0.42) RAD52RECQLGRM5
SCHEMBL14930325 0.63
SCHEMBL16286090 0.60 RAD52 (0.69) RAD52RECQLGRM5
SCHEMBL14925537 0.60 GAA (0.38)
SCHEMBL17088087 0.59 RAD52 (0.49) RAD52RECQLGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180071286-A1 HETEROARYL PYRIDONE AND AZA-PYRODINE COMPOUNDS GENENTECH, INC. (US) 2018-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180071286-A1 HETEROARYL PYRIDONE AND AZA-PYRODINE COMPOUNDS TYK2, BTK, PDXK RAD52 1050/4885RECQL 934/4885PTGDR2 728/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.