SCHEMBL19966566

SCHEMBL19966566

Cc1[nH]c2c(F)cc(-c3nc(Nc4ccc5c(n4)CCNC5)ncc3F)cc2c1C(C)C

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.63
CDK6 Q00534 20/20 0.63
CDK2 P24941 18/20 0.63
CDK1 P06493 4/20 0.63
CDK7 P50613 4/20 0.63
CDK9 P50750 4/20 0.63
CDK5 Q00535 3/20 0.61
CCNA2 P20248 4/20 0.59
CSF1R P07333 2/20 0.59
CCND3 P30281 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19966570 0.84 CDK4 (0.65) CDK4CDK6CDK2CDK1CDK7
SCHEMBL20356501 0.80 CDK4 (0.67) CDK4CDK6CDK2CDK1CDK7
SCHEMBL20356494 0.80 CDK4 (0.63) CDK4CDK6CDK2CDK1CDK7
SCHEMBL19966658 0.79 CDK6 (0.64) CDK4CDK6CDK2CDK1CDK7
SCHEMBL19966508 0.79 CDK4 (0.77) CDK4CDK6CDK2CDK1CDK7
SCHEMBL19966655 0.79 CDK6 (0.64) CDK4CDK6CDK2CDK1CDK9
SCHEMBL19966557 0.79 CDK4 (0.72) CDK4CDK6CDK2CDK1CDK7
SCHEMBL19966332 0.79 CDK6 (0.57) CDK4CDK6CDK2CDK1CDK7
SCHEMBL17477259 0.77 CDK4 (1.00) CDK4CDK6CDK2CDK1CDK7
SCHEMBL20548734 0.77 CDK4 (0.77) CDK4CDK6CDK2CDK1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045957-A1 CDK4/6 INHIBITOR AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed