SCHEMBL19966570

SCHEMBL19966570

CCN1CCc2nc(Nc3ncc(F)c(-c4cc(F)c5[nH]c(C)c(C(C)C)c5c4)n3)ccc2C1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.65
CCNE1 P24864 14/20 0.65
CDK1 P06493 14/20 0.65
CCNB1 P14635 13/20 0.65
CDK6 Q00534 10/20 0.58
CDK2 P24941 9/20 0.58
CDK9 P50750 4/20 0.55
CDK7 P50613 3/20 0.55
CCND3 P30281 3/20 0.55
CCNA2 P20248 2/20 0.55
CCNT1 O60563 2/20 0.54
CHEK1 O14757 1/20 0.54
JAK2 O60674 1/20 0.54
CHEK2 O96017 1/20 0.54
EGFR P00533 1/20 0.54
RAF1 P04049 1/20 0.54
NTRK1 P04629 1/20 0.54
PDGFRB P09619 1/20 0.54
SRC P12931 1/20 0.54
BRAF P15056 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19966566 0.84 CDK4 (0.63) CDK4CDK1CDK6CDK2CDK9
SCHEMBL19966656 0.82 CDK6 (0.60) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL19966451 0.82 CDK6 (0.64) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL19966547 0.82 CDK6 (0.48) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL19966510 0.81 CDK4 (0.79) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL19966556 0.79 CDK4 (0.72) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL19966325 0.79 CDK6 (0.61) CDK4CDK6CCND3
SCHEMBL17477262 0.79 CDK4 (1.00) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL18289076 0.78 CDK4 (1.00) CDK4CCNE1CDK1CCNB1CDK6
SCHEMBL18289326 0.78 CDK4 (1.00) CDK4CCNE1CDK1CCNB1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045957-A1 CDK4/6 INHIBITOR AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed