SCHEMBL19970854

SCHEMBL19970854

CCOP(=O)(Cc1ccc(COc2ccccc2N2CCN(Cc3ccc4nc(-c5ccc(C(F)(F)F)cc5)[nH]c4c3)CC2)cc1)OCC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.48
SLC2A1 P11166 2/20 0.47
GNRHR P30968 11/20 0.47
TACR2 P21452 1/20 0.47
HRH2 P25021 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
DRD4 P21917 1/20 0.41
PARP1 P09874 2/20 0.41
PARP6 Q2NL67 2/20 0.41
PARP2 Q9UGN5 2/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
HTR2A P28223 1/20 0.40
PARP3 Q9Y6F1 1/20 0.40
DGAT1 O75907 1/20 0.40
SOAT1 P35610 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19970850 0.94 GNRHR (0.47) MAOBSLC2A1GNRHRTACR2HRH2
SCHEMBL19982578 0.92 SLC2A1 (0.45) MAOBSLC2A1GNRHRTACR2HRH2
SCHEMBL19970889 0.89 SLC2A1 (0.44) MAOBSLC2A1GNRHRTACR2HRH2
SCHEMBL23843058 0.88 CHEK2 (0.43) SLC2A1DRD4DRD3DGAT1SOAT1
SCHEMBL19982561 0.87 SLC2A1 (0.46) MAOBSLC2A1GNRHRTACR2HRH2
SCHEMBL19970810 0.86 CHEK2 (0.41) SLC2A1DGAT1KCNH2
SCHEMBL19982610 0.85 SLC2A1 (0.42) SLC2A1DRD4DRD3HTR2AKCNH2
SCHEMBL19970888 0.84 GNRHR (0.41) MAOBSLC2A1GNRHRTACR2HRH2
SCHEMBL19970801 0.84 CHEK2 (0.43) SLC2A1DRD4DRD3DGAT1SOAT1
SCHEMBL19982564 0.82 SLC2A1 (0.42) SLC2A1DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3296297-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-21 EP disclosed