SCHEMBL19974536

SCHEMBL19974536

O=C(O)/C=C/C(=O)Nc1ccnc(-c2ccncc2)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.55
KDM4E B2RXH2 5/20 0.55
MAPT P10636 5/20 0.55
KMT2A Q03164 3/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
LPAR2 Q9HBW0 2/20 0.53
LPAR1 Q92633 1/20 0.53
LPAR3 Q9UBY5 2/20 0.50
CREBBP Q92793 1/20 0.49
PARP1 P09874 2/20 0.48
PARP15 Q460N3 2/20 0.48
PARP14 Q460N5 2/20 0.48
PARP10 Q53GL7 2/20 0.48
CNR1 P21554 1/20 0.47
TDP2 O95551 1/20 0.45
GAA P10253 1/20 0.45
THRB P10828 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
POLB P06746 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19974537 1.00 ALDH1A1 (0.55) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL23647318 0.90 ALDH1A1 (0.59) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL19974422 0.90 ALDH1A1 (0.59) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL19974201 0.86 NMT1 (0.60) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL19974204 0.86 NMT1 (0.60) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL19974429 0.85 ALDH1A1 (0.64) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL23647316 0.85 ALDH1A1 (0.64) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL11753292 0.82 CNR1 (0.54) ALDH1A1KDM4EKMT2ASMN1; SMN2CNR1
SCHEMBL19974155 0.82 LPAR2 (0.67) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL19974157 0.82 LPAR2 (0.67) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512602-A2 INHIBITORS OF HEAT SHOCK FACTORS AND USES THEREOF HSF Pharmaceuticals (CH) 2019-07-24 EP disclosed
WO-2018050656-A2 INHIBITORS OF HEAT SHOCK FACTORS AND USES THEREOF HSF PHARMACEUTICALS (CH) 2018-03-22 WO disclosed