SCHEMBL19974705

SCHEMBL19974705

O=C(Cc1ccccc1)Oc1cnc[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.46
CPA1 P15085 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TAAR1 Q96RJ0 2/20 0.44
HRH3 Q9Y5N1 1/20 0.44
PAM P19021 1/20 0.44
TSHR P16473 2/20 0.42
IDO1 P14902 1/20 0.41
UCHL1 P09936 1/20 0.41
USP5 P45974 1/20 0.41
USP4 Q13107 1/20 0.41
SENP1 Q9P0U3 1/20 0.41
CYP3A4 P08684 1/20 0.41
GABRA1 P14867 1/20 0.41
NFKB1 P19838 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10359891 0.79 KMT2A (0.52) MEN1KMT2ACPA1ALDH1A1MAPK1
SCHEMBL29020257 0.76 SMN1; SMN2 (0.50) CYP19A1KMT2ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL7279175 0.75 ALDH1A1 (0.39) MEN1KMT2ASMN1; SMN2ALDH1A1HRH3
SCHEMBL3961101 0.74
SCHEMBL19974645 0.72 MEN1 (0.38) MEN1KMT2ASMN1; SMN2ALDH1A1HRH3
SCHEMBL19974760 0.71 HRH3 (0.40) MEN1KMT2AALDH1A1HRH3TSHR
SCHEMBL538524 0.70 CYP19A1 (0.76) CYP19A1KMT2ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL10573912 0.70 MAPK1 (0.61) CYP19A1KMT2ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL2216126 0.70 CYP19A1 (0.69) CYP19A1KMT2ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL29020312 0.70 SMN1; SMN2 (0.55) CYP19A1KMT2ASMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512840-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS Tseng, Yufeng, Jane (US) 2019-07-24 EP disclosed
WO-2018053161-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS NATIONAL TAIWAN UNIVERSITY (TW) 2018-03-22 WO disclosed