SCHEMBL19975111

SCHEMBL19975111

CC(Cl)C(=O)Oc1cnc[nH]1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 1/20 0.38
GABRA1 P14867 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
GABRR1 P24046 1/20 0.38
GABRR2 P28476 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRB2 P47870 1/20 0.38
GABRA4 P48169 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
PMP22 Q01453 1/20 0.37
HRH3 Q9Y5N1 10/20 0.36
HRH4 Q9H3N8 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19974669 0.87 ELANE (0.38) HRH3HRH4MEN1KMT2A
SCHEMBL19975343 0.79 HRH3 (0.40) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL4605470 0.78 MEN1 (0.45) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL7158594 0.77
SCHEMBL3961101 0.75
SCHEMBL1331771 0.74 MEN1 (0.38) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL7449177 0.74 ALDH1A1 (0.40) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL13134162 0.71 KMT2A (0.36) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL19974661 0.70 MEN1 (0.41) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL13134160 0.69 MEN1 (0.40) ALDH1A1CYP3A4GABRA1TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512840-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS Tseng, Yufeng, Jane (US) 2019-07-24 EP disclosed
WO-2018053161-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS NATIONAL TAIWAN UNIVERSITY (TW) 2018-03-22 WO disclosed