SCHEMBL19979252

SCHEMBL19979252

CCOP(=O)(OCC)OC[C@H]1O[C@@H](n2cnc3c(=O)[nH]cnc32)C(C)(CO)C1O

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.51
ADORA3 P0DMS8 3/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
ALB P02768 1/20 0.42
MAPK1 P28482 1/20 0.42
TYMP P19971 4/20 0.41
GSK3A P49840 2/20 0.40
RPS6KA3 P51812 2/20 0.40
MAPK14 Q16539 2/20 0.40
IMPDH2 P12268 1/20 0.38
IMPDH1 P20839 1/20 0.38
STING1 Q86WV6 1/20 0.37
ADORA2A P29274 1/20 0.37
NT5E P21589 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19978970 0.92 P2RX3 (0.56) P2RX3ADORA3ALDH1A1LMNAALB
SCHEMBL22700214 0.85 HPGD (0.49) IMPDH2IMPDH1ADORA2ANT5E
SCHEMBL19974568 0.85 ADORA2A (0.55) P2RX3ALDH1A1ADORA2ANT5E
SCHEMBL19979029 0.81 ADORA2A (0.57) ADORA3LMNAADORA2ANT5E
SCHEMBL19974418 0.81 ADORA2A (0.57) ADORA3LMNAADORA2ANT5E
SCHEMBL19974575 0.79 ADORA2A (0.43) ADORA3ADORA2ANT5E
SCHEMBL15045893 0.75 ADORA2A (0.52) P2RX3ADORA3ALDH1A1LMNAALB
SCHEMBL13559257 0.73 ADORA2A (0.66) P2RX3ADORA3ALDH1A1LMNAALB
SCHEMBL12149438 0.73 ADORA2A (0.66) P2RX3ADORA3ALDH1A1LMNAALB
SCHEMBL13559231 0.73 ADORA2A (0.66) P2RX3ADORA3ALDH1A1LMNAALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512860-B1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC (CA) 2020-11-25 EP disclosed
WO-2018049534-A1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC. (CA) 2018-03-22 WO disclosed