SCHEMBL19980211

SCHEMBL19980211

CCCC/C=C(\N)C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 1/20 0.43
GRIK1 P39086 1/20 0.43
FAAH O00519 3/20 0.42
SOAT1 P35610 2/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
TSHR P16473 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CNR1 P21554 1/20 0.39
KDM4E B2RXH2 2/20 0.38
F7 P08709 1/20 0.38
F3 P13726 1/20 0.38
ALDH1A1 P00352 2/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29134998 1.00 EP300 (0.43) EP300GRIK1FAAHSOAT1MEN1
SCHEMBL5084408 0.91 EP300 (0.55) EP300FAAHSOAT1MEN1TP53
SCHEMBL639212 0.85
SCHEMBL11747745 0.85
SCHEMBL4280231 0.84 EP300 (0.52) EP300GRIK1FAAHSOAT1MEN1
Butane SCHEMBL6767216 0.83 GRIK1 (0.38) EP300GRIK1FAAHSOAT1MEN1
Hydrochloric Acid SCHEMBL6055071 0.83 GRIK1 (0.38) EP300GRIK1FAAHSOAT1MEN1
Chloromethane SCHEMBL18426109 0.81 GRIK1 (0.37) EP300GRIK1FAAHSOAT1MEN1
SCHEMBL180918 0.79 EP300 (0.42) EP300GRIK1FAAHSOAT1MEN1
SCHEMBL5831469 0.79 EP300 (0.47) EP300GRIK1FAAHSOAT1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3375780-B1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2020-06-03 EP disclosed
EP-3542193-A1 METHOD FOR MAKING OPHTHALMIC LENSES Novartis AG (CH) 2019-09-25 EP disclosed
US-20180141293-A1 METHOD FOR MAKING OPHTHALMIC LENSES ALCON INC. (CH) 2018-05-24 US disclosed
EP-2956452-B1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2018-03-21 EP disclosed