SCHEMBL19980669

SCHEMBL19980669

CC(=O)NC1CCC(CN2CCC(c3cn(-c4ccc(F)cc4C(=O)N(C)C(C)C)c4cnccc34)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.40
DRD3 P35462 6/20 0.40
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
OPRL1 P41146 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KCNH2 Q12809 1/20 0.36
DRD2 P14416 3/20 0.36
HRH2 P25021 1/20 0.35
ACKR3 P25106 1/20 0.34
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19972510 1.00 HTR2A (0.40) HTR2ADRD3OPRM1OPRK1OPRL1
SCHEMBL19972513 1.00 HTR2A (0.40) HTR2ADRD3OPRM1OPRK1OPRL1
SCHEMBL19972578 0.94 OPRM1 (0.38) HTR2ADRD3OPRM1OPRK1OPRL1
SCHEMBL19972669 0.94 OPRM1 (0.38) HTR2ADRD3OPRM1OPRK1OPRL1
SCHEMBL19972654 0.94 HTR2A (0.48) HTR2ADRD3DRD2
SCHEMBL19972657 0.94 HTR2A (0.48) HTR2ADRD3DRD2
SCHEMBL19972462 0.91 OPRM1 (0.41) OPRM1OPRK1OPRL1MEN1KMT2A
SCHEMBL30265628 0.91 OPRM1 (0.41) OPRM1OPRK1OPRL1MEN1KMT2A
SCHEMBL19972463 0.91 OPRM1 (0.41) OPRM1OPRK1OPRL1MEN1KMT2A
SCHEMBL30524094 0.91 OPRM1 (0.41) OPRM1OPRK1OPRL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118359610-A MENIN-MLL interaction inhibitors 生命医药有限责任公司 2024-07-19 CN disclosed
EP-4230627-A2 INHIBITORS OF THE MENIN-MLL INTERACTION Vitae Pharmaceuticals, LLC (US) 2023-08-23 EP disclosed
EP-3512850-B1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS LLC (US) 2023-04-12 EP disclosed
WO-2018053267-A1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS, INC. (US) 2018-03-22 WO disclosed