SCHEMBL19983077

SCHEMBL19983077

C[C@H](NC(=O)c1cccc(-n2cc(CN)nn2)c1)C(=O)COc1c(F)cc(CNC(=O)c2ccc(/N=N/c3ccc(N(C)C)cc3)cc2)cc1F

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 2/20 0.35
TSHR P16473 1/20 0.34
ALOX15 P16050 1/20 0.34
PTGS2 P35354 1/20 0.34
MIF P14174 2/20 0.33
TYMS P04818 1/20 0.33
KLKB1 P03952 1/20 0.33
KLK1 P06870 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983116 0.86 MEN1 (0.34)
SCHEMBL21152646 0.81 FOLH1 (0.35)
SCHEMBL21153288 0.76 ESRRA (0.37)
SCHEMBL21153247 0.75 CTSK (0.41)
SCHEMBL21153255 0.75 CTSK (0.41)
SCHEMBL19982920 0.74 CTSK (0.39)
SCHEMBL21113155 0.74 CTSK (0.39)
SCHEMBL19982922 0.74 CTSK (0.39)
SCHEMBL25658857 0.70 ESRRA (0.38)
SCHEMBL21153262 0.69 PRSS1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed