SCHEMBL19983233

SCHEMBL19983233

CN(C)c1ccc(/N=N/c2ccc(C(=O)NCc3cc(F)c(OCC(=O)CCCCCNC(=O)OC(C)(C)C)c(F)c3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 12/20 0.40
HDAC6 Q9UBN7 12/20 0.40
HDAC10 Q969S8 11/20 0.40
HDAC8 Q9BY41 10/20 0.40
HDAC2 Q92769 9/20 0.40
HDAC3 O15379 8/20 0.40
HDAC4 P56524 7/20 0.40
HDAC7 Q8WUI4 7/20 0.40
HDAC11 Q96DB2 7/20 0.40
HDAC9 Q9UKV0 7/20 0.40
HDAC5 Q9UQL6 7/20 0.40
LTA4H P09960 1/20 0.40
CYP3A4 P08684 1/20 0.39
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21152659 0.79 ALB (0.38) MAPT
SCHEMBL19983328 0.78 ESRRG (0.44) HDAC1HDAC6HDAC3CYP3A4
SCHEMBL25660999 0.77 ALB (0.35) KDM4EALDH1A1MAPT
SCHEMBL25658966 0.75 TDP1 (0.39) KDM4EMAPTRAB9A
SCHEMBL19983116 0.75 MEN1 (0.34) MAPT
SCHEMBL19983300 0.74 KDM4E (0.56) HDAC1HDAC6HDAC10HDAC8HDAC2
SCHEMBL19982963 0.74 CYP3A4 (0.49) CYP3A4KDM4E
SCHEMBL21152665 0.73 ALB (0.39)
SCHEMBL17623614 0.71 HDAC1 (0.61) HDAC1HDAC6HDAC10HDAC8HDAC2
SCHEMBL19983069 0.71 CYP3A4 (0.46) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed