SCHEMBL19983069

SCHEMBL19983069

CC(C)(C)OC(=O)NCCCCCC(=O)COc1c(F)ccc(F)c1F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
CA1 P00915 6/20 0.44
CA2 P00918 6/20 0.44
CA12 O43570 5/20 0.44
CA9 Q16790 5/20 0.44
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
DRD2 P14416 2/20 0.40
CTSK P43235 1/20 0.39
PLK1 P53350 1/20 0.39
TPSAB1 Q15661 1/20 0.39
TPSD1 Q9BZJ3 1/20 0.39
TPSG1 Q9NRR2 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19982963 0.90 CYP3A4 (0.49) CYP3A4TDP1CA1CA2CA12
SCHEMBL19983252 0.76 CYP3A4 (0.50) CYP3A4TDP1CA1CA2CA12
SCHEMBL4956882 0.76 TDP1 (0.50) CYP3A4TDP1CA1CA2CA12
SCHEMBL19983124 0.76 CTSK (0.48) CTSK
SCHEMBL19983325 0.75 CTSK (0.75) TDP1CTSKPOLB
SCHEMBL30958391 0.74 TDP1 (0.68) CYP3A4TDP1CA1CA2CA12
SCHEMBL11982402 0.74 CA1 (0.46) TDP1CA1CA2CA12CA9
SCHEMBL8634314 0.73 TDP1 (0.55) CYP3A4TDP1CA1CA2CA12
SCHEMBL11900877 0.72 CA1 (0.47) TDP1CA1CA2CA12CA9
SCHEMBL12634724 0.72 TDP1 (0.45) TDP1CA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed